Not available in the U.S.
Mechanism of action: Ethacizine ballicule
What it isClass IC antiarrhythmic used in Russia.
Why this oneAvailable where other class IC agents are not.
What limits itThe CAST proarrhythmia concern applies to the class. Not US-approved.
Molecular structure: Ethacizine
FDA-approved for
- cardiac arrhythmias (non-US)
Off-label
- arrhythmias (approved in Russia)
Principal riskThe CAST proarrhythmia concern applies to the class
Classes and tags
Clinical profile
Therapeutic safety burden3 / 4
Overdose danger3 / 4
QT / Torsades0 / 4
Direct muscarinic antagonism0 / 4
Defining liabilityProarrhythmia, conduction block and impaired myocardial contractility
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