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Aluminum hydroxide

AMPHOJEL

Pronunciation: a-LOO-mi-num hye-DROX-ide

Aluminum hydroxide ballicule: receptor binding, kinetics and half-life diagram
Mechanism of action: Aluminum hydroxide ballicule

What it isAluminum antacid that neutralizes gastric acid and binds phosphate; short-term dyspepsia and refractory hyperphosphatemia.

Why this oneIts phosphate binding once made it useful in renal failure, but safer nonaluminum binders have largely replaced it.

What limits itIt binds quinolones, tetracyclines and levothyroxine; constipation and neurotoxic accumulation make chronic use unsafe in kidney disease.

Aluminum hydroxide molecular structure (skeletal formula)
Molecular structure: Aluminum hydroxide

Available strengths

NO BOXED WARNINGS

Principal riskNo FDA boxed warning.

Classes and tags

Clinical profile

Therapeutic safety burden0 / 4
Sedation liability0 / 4
Direct muscarinic antagonism0 / 4
Embryofetal risk1 / 4

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